Fol. Biol. 2016, 62, 167-174

https://doi.org/10.14712/fb2016062040167

Comparison of the Radiosensitizing Effect of ATR, ATM and DNA-PK Kinase Inhibitors on Cervical Carcinoma Cells

Jiřina Vávrová1, L. Zárybnická1, P. Jošt2, A. Tichý1, M. Řezáčová3, Z. Šinkorová1, J. Pejchal1

1Department of Radiobiology, Faculty of Military Health Sciences, Hradec Králové, University of Defence Brno, Czech Republic
2Centre of Advanced Studies, Faculty of Military Health Sciences, Hradec Králové, University of Defence Brno, Czech Republic
3Institute of Medical Biochemistry, Charles University Prague, Faculty of Medicine in Hradec Králové, Czech Republic

Received November 2015
Accepted April 2016

Crossref Cited-by Linking

  • Kopa Paulina, Macieja Anna, Pastwa Elzbieta, Majsterek Ireneusz, Poplawski Tomasz: DNA double-strand breaks repair inhibitors potentiates the combined effect of VP-16 and CDDP in human colorectal adenocarcinoma (LoVo) cells. Mol Biol Rep 2021, 48, 709. <https://doi.org/10.1007/s11033-020-06124-9>
  • Faulhaber Eva-Maria, Jost Tina, Symank Julia, Scheper Julian, Bürkel Felix, Fietkau Rainer, Hecht Markus, Distel Luitpold V.: Kinase Inhibitors of DNA-PK, ATM and ATR in Combination with Ionizing Radiation Can Increase Tumor Cell Death in HNSCC Cells While Sparing Normal Tissue Cells. Genes 2021, 12, 925. <https://doi.org/10.3390/genes12060925>
  • Medová Michaela, Medo Matú\u0161, Hovhannisyan Lusine, Muñoz-Maldonado Carmen, Aebersold Daniel M., Zimmer Yitzhak: DNA-PK in human malignant disorders: Mechanisms and implications for pharmacological interventions. Pharmacology & Therapeutics 2020, 215, 107617. <https://doi.org/10.1016/j.pharmthera.2020.107617>
  • Wong Way Wua, Jackson Rosanna K., Liew Lydia P., Dickson Benjamin D., Cheng Gary J., Lipert Barbara, Gu Yongchuan, Hunter Francis W., Wilson William R., Hay Michael P.: Hypoxia-selective radiosensitisation by SN38023, a bioreductive prodrug of DNA-dependent protein kinase inhibitor IC87361. Biochemical Pharmacology 2019, 169, 113641. <https://doi.org/10.1016/j.bcp.2019.113641>
  • Lee Tet Woo, Wong Way Wua, Dickson Benjamin D., Lipert Barbara, Cheng Gary J., Hunter Francis W., Hay Michael P., Wilson William R.: Radiosensitization of head and neck squamous cell carcinoma lines by DNA-PK inhibitors is more effective than PARP-1 inhibition and is enhanced by SLFN11 and hypoxia. International Journal of Radiation Biology 2019, 95, 1597. <https://doi.org/10.1080/09553002.2019.1664787>
  • Cossar L.H., Schache A.G., Risk J.M., Sacco J.J., Jones N.J., Lord R.: Modulating the DNA Damage Response to Improve Treatment Response in Cervical Cancer. Clinical Oncology 2017, 29, 626. <https://doi.org/10.1016/j.clon.2017.03.002>
Crossref Cited-by Linking logo